Bilastine is an advanced second-generation antihistamine that has garnered attention in the pharmaceutical world for its effectiveness in treating allergic conditions without causing drowsiness. With allergic disorders becoming increasingly prevalent, the demand for safer and more effective antihistamines is growing. Among the notable manufacturers of Bilastine API, Valence Labs stands out as a trusted name in the Indian pharmaceutical API industry.
In this blog, we’ll explore everything you need to know about Bilastine, including its uses, benefits, potential side effects, and why Valence Labs is your ideal partner for high-quality Bilastine API.
Bilastine is a non-sedating antihistamine used primarily to treat symptoms of allergic rhinitis and chronic urticaria (hives). It works by selectively inhibiting peripheral histamine H1 receptors, which helps block the release of histamines responsible for allergy symptoms.
Its is recognized for its fast onset of action, prolonged effect, and minimal side effects compared to first-generation antihistamines like diphenhydramine and chlorpheniramine.
Bilastine is prescribed for the management of:
A condition triggered by allergens such as dust, pollen, and pet dander. Symptoms include:
A long-term skin condition marked by:
Its provides quick relief from symptoms caused by environmental changes, pollen, or climate shifts, especially during spring and fall.
Unlike traditional antihistamines, Its does not cross the blood-brain barrier significantly, making it less likely to cause drowsiness. This allows patients to go about daily activities without impairment.
Bilastine has a long half-life of around 14–15 hours, ensuring 24-hour symptom control with just a single dose daily.
Onset of action typically occurs within one hour, providing fast relief from allergy symptoms.
Its is metabolized minimally by the liver, resulting in fewer interactions with other medications—especially important for patients on multiple drugs.
Clinical trials have shown that Bilastine is safe for extended use in treating chronic allergies.
Although generally well tolerated, some patients may experience minor side effects, including:
These symptoms are usually mild and resolve without intervention. However, serious side effects are extremely rare.Â
At Valence Labs, we are proud to be among the leading manufacturers and suppliers of Bilastine API in India. Our commitment to high-quality production, GMP-certified facilities, and strict quality control makes us a preferred partner for pharmaceutical companies across the globe.
Whether you’re a formulation company or a global pharma distributor, partnering with Valence Labs ensures you receive consistent, high-quality API to support your end-products.
Feature |
Bilastine | Cetirizine | Loratadine |
Drowsiness |
Minimal | Mild to Moderate | Mild |
Onset of Action |
~1 Hour | ~1 Hour | 1–3 Hours |
Half-Life | ~14 Hours | ~8 Hours |
~8 Hours |
Frequency | Once Daily | Once Daily |
Once Daily |
Food Interaction | Yes (absorption reduced) | No |
No |
Bilastine has revolutionized allergy treatment by offering a non-sedating, effective, and safe option for long-term relief. With the rising prevalence of allergic conditions, its demand is only expected to grow. If you are looking for a reliable Bilastine API manufacturer, look no further than Valence Labs.
We are committed to providing the highest quality APIs with integrity, precision, and innovation. Valence Labs today to discuss your bulk API requirements for other pharmaceutical products.
Contact Valence labs, if you want to get any details regarding Bilastine Or any other details regarding our company.